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カタログ番号	製品名	別名	ターゲット
T9744	MP07-66		Phosphatase
	MP07-66 is a novel FTY720-analog devoid of immunosuppressive effects leads to the reactivation of PP2A, which in turn triggers apoptosis of CLL cells.		Phosphatase
T60022	Aromatase-IN-2		Others
	Aromatase-IN-2 has anti-inflammatory, antitumor and antiasthmatic effects.		Others
T13111	Tegadifur	40497S,FD 1	Others
	Tegadifur (40497S) is an orally available antitumor compound with antimetabolic effects, often used with uracil and in the treatment of rectal adenocarcinoma.		Others
T9992	SphK1&2-IN-1		S1P Receptor
	SphK1&2-IN-1 is a sphingosine kinase inhibitor with anti-inflammatory, antitumor and hemostatic effects.		S1P Receptor
T5845	7ACC1	DEAC,Coumarin D 1421,7-(Diethylamino)coumarin-3-carboxylic acid,D 1421	Monocarboxylate transporter
	7ACC1 (D 142) selectively affects a single part of the MCT symporter translocation cycle, leading to strict inhibition of lactate influx. This singular activity is associated with antitumor effects less prone to resistan...		Monocarboxylate transporter
T23911	CPS-11	CPS11,CPS 11,N-(Hydroxymethyl)thalidomide	Dehydrogenase , NF-κB , Reactive Oxygen Species
	CPS-11 (N-(Hydroxymethyl)thalidomide) is a Thalidomide analogue that has significant antitumor activity and exhibits a wider range of activity and highly potent effects on the MM (multiple myeloma) cell line.		Dehydrogenase , NF-κB , Reactive Oxygen Species
T72551	Antitumor agent-87
	Antitumor agent-87 is a potent compound with antitumoral activity, demonstrating a high affinity for CYP1A1, evidenced by a K i value of 0.23 µM. It exhibits antiproliferative effects and induces cell cycle arrest at the...
T16551	Pladienolide B		Apoptosis
	Pladienolide B is a potent spliceosome inhibitor, a macrolide isolated from Streptomyces obtusususus Mer-12, which targets the SF3B1 subunit of the spliceosome.Pladienolide B exerts its antitumor effects by inhibiting pr...		Apoptosis
TNU0425	2’-Deoxy-2’-fluoro-β-D-arabinocytidine hydrochloride		DNA Methyltransferase
	2’-Deoxy-2’-fluoro-β-D-arabinocytidine hydrochloride is a cytosine nucleoside analog with inhibitory effects on DNA methyltransferase , with potential antimetabolic and antitumor activity.		DNA Methyltransferase
T13174	TMPyP4 tosylate	TMP 1363	DNA/RNA Synthesis , Telomerase
	TMPyP4 tosylate (TMP 1363) is a quadruplex-specific ligand and is a telomerase inhibitor with antitumor effects in osteosarcoma cell lines.		DNA/RNA Synthesis , Telomerase
T60082	HDAC-IN-40		HDAC
	HDAC-IN-40 is a potent alkoxyamide-based HDAC inhibitor with Ki of 60 nM and 30 nM for HDAC2 and HDAC6, respectively. HDAC-IN-40 had antitumor effects		HDAC
T76780	Onartuzumab	RG-3638,PRO-14396,MetMAb	c-Met/HGFR
	Onartuzumab (MetMAb) is a humanized anti-tyrosine kinase c-MET monovalent monoclonal antibody.Onartuzumab has antitumor activity with inhibitory effects on HGF binding, receptor phosphorylation, and signal transduction.		c-Met/HGFR
T76761	Olaratumab	LY3012207,IMC-3G3	PDGFR
	Olaratumab(IMC-3G3) is a human monoclonal IgG1 antibody against platelet-derived growth factor receptor alpha (PDGFRα), which has antitumor effects and can be used to study advanced soft tissue sarcomas.		PDGFR
T5523	Imidazole ketone erastin	IKE	Ferroptosis
	Imidazole ketone erastin (IKE) is an iron death inducer with inhibitory effects on system Xc-cystine/glutamate transporter proteins. Imidazole ketone erastin has antitumor activity and induces glutathione depletion and l...		Ferroptosis
T77493	Murlentamab	3C23K,GM102	Others
	Murlentamab (GM102) is a humanized anti-AMhRII antibody. Murlentama has potential antitumor activity that induces macrophage-mediated antitumor-dependent cell-mediated cytotoxic effects (ADCC). Murl can stimulate the pro...		Others
T50071	Xanthine dehydrogenase Inhibitor 1		Others
	5-amino-1-[4-(trifluoromethyl)phenyl]-1H-pyrazole-4-carbonitrile is a compound used as a molecular structural unit and is considered to be an inhibitor of enzymes such as COX-2, 5-LOX, etc., and possesses a wide range of...		Others
T77437	Telisotuzumab	ABT-700,Mab-224G11	c-Met/HGFR
	Telisotuzumab(ABT-700) is a humanized recombinant antibody targeting the therapeutic hepatocyte growth factor receptor (MET) with high affinity for c-Met.Telisotuzumab has inhibitory effects on c-Met signaling and antitu...		c-Met/HGFR
T60680	Tegaserod		5-HT Receptor
	Tegaserod is an orally available 5-HT4R agonist and 5-HT2B receptor antagonist with inhibitory effects on various 5-hydroxytryptamine receptors. Tegaserod has antitumor activity and is used in the treatment of irritable ...		5-HT Receptor
T68090	Laprafylline		Others
	Laprafylline is a xanthine compound with inhibitory effects on bronchoconstriction in vivo and antitumor activity.Laprafylline acts as a competitive serotonergic antagonist at low concentrations, and inhibits constrictio...		Others
T62714	IRAK4-IN-20	BAY-1834845	IRAK
	IRAK4-IN-20 is a potent and orally active IRAK4 inhibitor (IC50:3.55 nM). IRAK4-IN-20, which has anti-inflammatory, antitumor and anticancer effects, is often used to treat acute respiratory distress syndrome (ARDS).		IRAK
T36488	LYG-202	LYG202,LYG 202	Apoptosis , ROS
	LYG-202 is a novel flavonoid with piperazine substitution and antitumor effects in vivo and in vitro.LYG-202 induced apoptosis in MCF-7, MDA-MB-231, and MDA-MB-435 cells, and increased intracellular ROS production.		Apoptosis , ROS
T68405L	KW-2450 Formate		Tyrosinase
	KW-2450 Formate is an IGF-1R/IR tyrosine kinase inhibitor with antitumor effects that acts through inhibition of Aurora A and B kinases.KW-2450 Formate inhibits the growth of TNBC xenografts and induces tetraploid accumu...		Tyrosinase
T76758	Rilotumumab	AMG 102	c-Met/HGFR
	Rilotumumab (AMG 102) is a monoclonal antibody targeting hepatocyte growth factor that inhibits HGF/ MET-driven signaling. Rilotumumab has antitumor effects and can be used to study castration-resistant prostate cancer (...		c-Met/HGFR
T69534	Zongertinib	BI 764532,BI 1810631	Tyrosine Kinases , HER
	Zongertinib is a human HER2-selective tyrosine kinase inhibitor, a novel TK that is highly selective for covalent binding to the HER2 tyrosine kinase domain (TKD).Zongertinib exhibits antitumor activity with inhibitory e...		Tyrosine Kinases , HER
TQ0181	Resatorvid	CLI-095,TAK-242	TNF , TLR , Autophagy , Interleukin
	Resatorvid (TAK-242) is a selective inhibitor of Toll-like receptor 4 (TLR4). Resatorvid binds directly to Cys747 and prevents TLR4 from binding to TIRAP, thereby blocking downstream signaling. Resatorvid has antitumor a...		TNF , TLR , Autophagy , Interleukin
T16156	MT 63-78		Apoptosis , AMPK , mTOR
	MT 63-78 is a specific and effective direct AMPK activator (EC50: 25 μM). MT 63-78 blocks prostate cancer growth by inhibiting the lipogenesis and mTORC1 pathways. MT 63-78 has antitumor effects. MT 63–78 also causes cel...		Apoptosis , AMPK , mTOR
T76941	Carotuximab	DE-122,TRC105	TGF-beta/Smad , Immunology/Inflammation related
	Carotuximab (DE-122) is a novel endocholine antibody with strong antiangiogenic and anti-inflammatory activity. Carotuximab blocks endothelial glycoprotein (CD105) and its downstream Smad signaling pathway. Carotuximab h...		TGF-beta/Smad , Immunology/Inflammation related
T27392	FT001		Epigenetic Reader Domain
	FT001 is a potent, selective and orally available inhibitor of BET Bromodomain with antitumor activity. FT001 inhibited the expression of MYC with the IC50 value of 0.46 μM). FT001 has potent antiproliferative effects ag...		Epigenetic Reader Domain
T4409	Gilteritinib	ASP2215	FLT , TAM Receptor , c-Kit
	Gilteritinib (ASP2215) is a potent inhibitor at the FMS-related tyrosine kinase 3 (FLT3) and AXL tyrosine kinase receptors (IC50 = 0.29 nM and <1 nM, respectively). In preClinicalal studies, gilteritinib showed strong an...		FLT , TAM Receptor , c-Kit
TP1592L	C-Reactive Protein (CRP) 174-185 acetate	C-Reactive Protein (CRP) 174-185 acetate(160369-86-8 free base)	Others
	C-Reactive Protein (CRP) 174-185 acetate is an acute phase serum protein synthesized in response to inflammatory cytokines, produces antitumor effects in animals. The fragment CRP (174-185) (RS-83277) shows similar activ...		Others
T61932	Nesuparib	JPI-547/OCN-201	PARP , Wnt/beta-catenin
	Nesuparib (JPI-547/OCN-201) is a potent PARP inhibitor with inhibitory effects on PARP and TNKS1.Nesuparib has antitumor activity and can be used in the treatment of tumors, endocrine and metabolic disorders, genitourina...		PARP , Wnt/beta-catenin
TF0106	Cholesteryl Hemisuccinate Tris Salt		Apoptosis
	Cholesteryl Hemisuccinate Tris Salt is an acidic cholesteryl ester with hepatoprotective and anticancer activity.Cholesteryl hemisuccinate is a membrane stabilizer in dipalmitoylphosphatidylcholine liposomes containing C...		Apoptosis
T77651	Tubulin polymerization-IN-47		Microtubule Associated
	Tubulin polymerization-IN-47 is a tubulin polymerization inhibitor and mitotic inhibitor with antitumor activity and inhibitory effects on neuroblastoma cancer cell proliferation, with IC50s of 7 and 12 nM for Chp-134 an...		Microtubule Associated
T36953	Naphthofluorescein	Naphthafluorescein	HIF
	Naphthofluorescein （Naphthafluorescein） is a Mint3 inhibitor with potential antitumor and anti-inflammatory activities, inhibits the interaction between HIF-1 and Mint3, inhibits Mint3-dependent HIF-1 activity, and inhib...		HIF
T60231	N-[2-nitro-4-(trifluoromethyl)phenyl]piperazine		Others
	N-[2-nitro-4-(trifluoromethyl)phenyl]piperazine is a biologically active compound belonging to the piperazine group. It is an important synthetic intermediate used in the preparation of a wide range of drugs, agrochemica...		Others
T3317	SZL P1-41		Apoptosis , Others , E1/E2/E3 Enzyme
	SZL P1-41, a skp2 inhibitor, can prevent assembly of Skp2-Skp1 complexes. It selectively suppresses Skp2 SCF E3 ligase activity but exhibits no effect on the activity of other SCF complexes. It also inhibits Skp2-mediate...		Apoptosis , Others , E1/E2/E3 Enzyme
T50100	3-hydroxy-3-phenylpentanamide		Others
	3-hydroxy-3-phenylpentanamide is a chiral compound belonging to the class of beta-hydroxyamides. In neurology, it has been shown to have neuroprotective effects against ischemic brain injury and cerebral hemorrhage. In p...		Others
T17731L	CL2A-SN-38 DCA 1279680-68-0(free base)		Others
	CL2A-SN-38 is a drug-linker conjugate composed of a potent a DNA Topoisomerase I inhibitor SN-38 and a linker CL2A to make antibody drug conjugate (ADC).. CL2A-SN-38 is composed of a potent a DNA Topoisomerase I inhibito...		Others
T36493	CMLD-2		Apoptosis , HuR
	CMLD-2 is an inhibitor of HuR-ARE interaction (Ki: 350 nM) that competitively binds HuR protein and disrupts its interaction with adenine element-rich (ARE) mRNA targets.CMLD-2 induces apoptosis and exhibits antitumor ef...		Apoptosis , HuR
T27369	FR 901537	FR901537,FR-901537
	FR 901537 is a new aromatase inhibitor with antitumor effects.
T12037	Mifamurtide	L-MTP-PE,MTP-PE,CGP 19835	Others
	Mifamurtide is a drug against osteosarcoma, is an immunomodulator with antitumor effects.		Others
T23633	Adechlorin
	Adechlorin is a synergistic antitumor and/or antiviral antibiotic. It potentiates the effects of other antitumor or antiviral compounds through the inhibition of key enzymes.
T30837	Cgp 47645	Leflutrozole,Cgp-47645,Cgp47645
	CGP 47645 (Leflurozole) is an oral active non-steroidal aromatase inhibitor and antitumor agent with anti-tumor and endocrine effects.
T30768	CB-403	UNII-4V9Q0C88UK,CB403,CB 403
	CB-403 is a cinnamaldehyde derivative that has antitumor effects by blocking cell cycle progression in the G2/M phase.
T4310L	Prexasertib lactate hydrate	Prexasertib monolactate monohydrate,LY-2606368,LY 2606368,LY2606368,Prexasertib monolactate monohydrate salt
	Prexasertib is an effective and selective Chk1/Chk2 inhibitor. Prexasertib causes Replication Catastrophe and Antitumor Effects through CHK1-Dependent Mechanisms.
T24813	SOMG-833 HCl	SOMG833 Hydrochloride,SOMG-833 Hydrochloride,SOMG 833 HCl,SOMG 833 Hydrochloride,SOMG833 HCl
	SOMG-833 HCl is a selective inhibitor of c-MET. It acts by blocking c-MET dependent neoplastic effects and exerting antitumor activity.
T11595	IACS-8779		Others
			Others
T68569	Aristoforin
	Aristoforin is a SIRT1 and SIRT2 inhibitor that induces cell cycle arrest, shows potent antitumor effects, and inhibits lymphangiogenesis in vivo.
T61806	Antitumor agent-44
	Antitumor agent-44 (Compound 5n) elicits potent antitumor effects by inducing disruption of mitochondrial homeostasis, cell cycle arrest, and apoptosis in human adenocarcinoma cells. Moreover, Antitumor agent-44 demonstr...
T72575	Antitumor agent-90
	Antitumor Agent-90 exhibits cytotoxic effects against PC 14 and MKN 45 cells, indicating its potential utility in cancer research.

Compounds

Synonym: DEAC,Coumarin D 1421,7-(Diethylamino)coumarin-3-carboxylic acid,D 1421

Target: Monocarboxylate transporter

CPS-11

T23911

Synonym: CPS11,CPS 11,N-(Hydroxymethyl)thalidomide

Target: Dehydrogenase, NF-κB, Reactive Oxygen Species

2’-Deoxy-2’-fluoro-β-D-arabinocytidine hydrochloride

TNU0425

Synonym:

Target: DNA Methyltransferase

TMPyP4 tosylate

T13174

Synonym: TMP 1363

Target: DNA/RNA Synthesis, Telomerase

Synonym: RG-3638,PRO-14396,MetMAb

Target: c-Met/HGFR

Olaratumab

T76761

Synonym: LY3012207,IMC-3G3

Target: PDGFR

Imidazole ketone erastin

Xanthine dehydrogenase Inhibitor 1

Synonym: ABT-700,Mab-224G11

Target: 5-HT Receptor

Synonym: LYG202,LYG 202

Target: Apoptosis, ROS

Synonym: BI 764532,BI 1810631

Target: Tyrosine Kinases, HER

Resatorvid

TQ0181

Synonym: CLI-095,TAK-242

Target: TNF, TLR, Autophagy, Interleukin

MT 63-78

T16156

Synonym:

Target: Apoptosis, AMPK, mTOR

Carotuximab

T76941

Synonym: DE-122,TRC105

Target: TGF-beta/Smad, Immunology/Inflammation related

FT001

T27392

Synonym:

Target: Epigenetic Reader Domain

Gilteritinib

T4409

Synonym: ASP2215

Target: FLT, TAM Receptor, c-Kit

C-Reactive Protein (CRP) 174-185 acetate

TP1592L

Synonym: C-Reactive Protein (CRP) 174-185 acetate(160369-86-8 free base)

Target: Others

Nesuparib

T61932

Synonym: JPI-547/OCN-201

Target: PARP, Wnt/beta-catenin

Cholesteryl Hemisuccinate Tris Salt

TF0106

Synonym:

Target: Apoptosis

Tubulin polymerization-IN-47

T77651

Synonym:

Target: Microtubule Associated

Naphthofluorescein

T36953

Synonym: Naphthafluorescein

Target: HIF

N-[2-nitro-4-(trifluoromethyl)phenyl]piperazine

Target: Apoptosis, Others, E1/E2/E3 Enzyme

3-hydroxy-3-phenylpentanamide

T50100

Synonym:

Target: Others

CL2A-SN-38 DCA 1279680-68-0(free base)

Target: Apoptosis, HuR

FR 901537

T27369

Synonym: FR901537,FR-901537

Target:

Mifamurtide

T12037

Synonym: L-MTP-PE,MTP-PE,CGP 19835

Synonym: Leflutrozole,Cgp-47645,Cgp47645

Target:

CB-403

T30768

Synonym: UNII-4V9Q0C88UK,CB403,CB 403

Target:

Prexasertib lactate hydrate

T4310L

Synonym: Prexasertib monolactate monohydrate,LY-2606368,LY 2606368,LY2606368,Prexasertib monolactate monohydrate salt

Target:

SOMG-833 HCl

T24813

Synonym: SOMG833 Hydrochloride,SOMG-833 Hydrochloride,SOMG 833 HCl,SOMG 833 Hydrochloride,SOMG833 HCl

カタログ番号	製品名	別名	ターゲット
TMS1743	Salvigenin		MAO , Autophagy , ROS Kinase
	Salvigenin is a potent hMAO-A inhibitor, has neuroprotective, antitumor and immunomodulatory effects.		MAO , Autophagy , ROS Kinase
TN6097	Girinimbine	Girinimbin	Apoptosis , Antioxidant , Antibacterial
	Girinimbine (Girinimbin) is a carbazole alkaloid isolated from the plants M. koenigii, M. koenigii and Murraya koenigii.Girinimbine has a wide range of biological effects, including apoptosis, antitrypanosomal, antiplate...		Apoptosis , Antioxidant , Antibacterial
T12971	Solanidine		Others
	Solanidine is a cholestane alkaloid isolated from potato species with antitumor effects. Solanidine inhibits proliferation.		Others
T19768	γ-Tocotrienol	gamma Tocotrienol,gammaTocotrienol,gamma-Tocotrienol,D-gamma-Tocotrienol,Plastochromanol	Others
	γ-Tocotrienol (Plastochromanol) is one of the four types of tocotrienol, a type of vitamin E. Itl is also a radioprotector, antioxidant. It shows antitumor and antihypertensive effects in vivo.		Others
T13350	Wushanicaritin		Others
	Wushanicaritin is a natural product isolated from the traditional Chinese medicine Epimedium plants, with antitumor effects and anti-inflammatory property.		Others
T38815	Millepachine		Apoptosis
	Millepachine is a natural product found in the Chinese herbal medicine with strong antitumor effects against numerous human cancer cells.		Apoptosis
T5S1607	Morusin	Mulberrochromene	NF-κB , Antibacterial , STAT
	1. Morusin (Mulberrochromene) possesses antitumor effects of cell lines including HT-29, A549, MCF-7, and MDA-MB-231, through suppressing STAT3 and NFκB attenuation mediated apoptosis induction. 2. Morusin possesses anti...		NF-κB , Antibacterial , STAT
TN6963	Hentriacontane		NF-κB
	Hentriacontane is a natural product.		NF-κB
TN2326	(Z)-Butylidenephthalide	(Z)-3-Butylidenephthalide	Glucosidase
	(Z)-Butylidenephthalide ((Z)-3-Butylidenephthalide) has antitumor and hypoglycemic effects, and can effectively inhibit the tumor growth of glioma and inhibit R-glucosidase activity.		Glucosidase
TN1148	Isopsoralenoside		Estrogen Receptor/ERR , Estrogen/progestogen Receptor , Antibacterial
	Isopsoralenoside shows estrogen-like, osteoblastic proliferation accelerating, antitumor, and antibacterial effects.
T5771	Hypocrellin A		Antibacterial , PKC , Parasite
	Hypocrellin A is PKC inhibitor, has light-induced antitumor,antifungal and antiviral activities, it also exerts immunomodulatory effects on MHC-restricted presentation of antigen.		Antibacterial , PKC , Parasite
T3408	Syringin	Lilacin,Syringoside,eleutheroside-b,Methoxyconiferine	NOS , Autophagy
	Syringin (eleutheroside-b) is a compound with antitumor, antiproliferative, immunomodulatory and platelet aggregation inhibiting effects.		NOS , Autophagy
T3386	Kaempferitrin	Lespedin,Kaempferol,Lespenephryl,Lespenefril,Kaempferol 3,7-dirhamnoside	cell cycle arrest , Glucokinase , IGF-1R
	Kaempferitrin (Lespenephryl) has antidepressant-like effect related to the serotonergic system, principally 5-HT1A. Kaempferitrin exerts cytotoxic and antitumor effects against HeLa cells. Kaempferitrin stimulates glucos...		cell cycle arrest , Glucokinase , IGF-1R
TN1008	Psoralenoside		CaMK , Calcium Channel , Histamine Receptor
	Psoralenoside is a natural product isolated from the fruits of Psoralea corylifolia, shows estrogen-like activity, osteoblastic proliferation accelerating activity, antitumor effects and antibacterial activity.		CaMK , Calcium Channel , Histamine Receptor
T25192	Butyrolactone I	Olomoucin	CDK
	Butyrolactone I (Olomoucin) is an ATP-competitive inhibitor of CDK and cdc2 kinase family. Butyrolactone I shows antitumor effects in non-small cell lung, small cell lung, and prostate cancer cell lines.		CDK
TN1130	Yadanziolide A		Antiviral
	Yadanziolide A is a natural product isolated from the cultivated dry seeds of Brucea javanica, has strong antiviral activities with IC50 of 5.5 μM against tobacco mosaic virus. Yadanziolide A shows significant antitumor ...		Antiviral
T2S0712	Sinigrin	Allylglucosinolate,2-Propenylglucosinolate	Others , Antioxidant
	Sinigrin is the major thioglucoside in Cruciferae with anti-adipogenic properties. It was used as reference material in the isolation and characterization procedure of mustard oleoresins.Sinigrin has potent antioxidant, ...		Others , Antioxidant
T6S0052	Chelerythrine	Toddalin,Broussonpapyrine,Cheleritrine	Apoptosis , BCL , PKC , Autophagy
	1. Chelerythrine (Broussonpapyrine) may have antimanic effect . 2. Chelerythrine can inhibit telomerase activity. 3. Chelerythrine is a well-known protein kinase C inhibitor . 4. Chelerythrine has potential antiprolifera...		Apoptosis , BCL , PKC , Autophagy
T7918	2-Amino-2-dichlorobenzophenone		Others
	2-Amino-2-dichlorobenzophenone is an aromatic natural compound that has been used to study the effects of various compounds on cell metabolism, protein synthesis and enzyme activity. It has also been used in the synthesi...		Others
T4S1999	Valepotriate	Valtrate	Apoptosis , HIV Protease
	Valepotriate (Valtrate) fraction can have sedative effects and affect behavioral parameters related to recognition memory. Valepotriates, a new class of cytotoxic and antitumor agents, they are very potent cytotoxic agen...		Apoptosis , HIV Protease
T2795	Amygdalin	Laetrile	Others
	Amygdalin (Laetrile) has antifibrotic, antitumor, anti-inflammatory and analgesic effects, amygdalin joint HSYA could inhibit the degeneration of the endplate chondrocytes derived from intervertebral discs of rats induce...		Others
T3822	Bellidifolin	Bellidifoline,Bellidifolium	Others , HIV Protease
	Bellidifolin (Bellidifoline) has anti-oxidation, hepatoprotective, anti-inflammatory and antitumor actions, it may contribute to the protective effects associated with nerve injury initiated by hypoxia by mechanisms rela...		Others , HIV Protease
TN1969	N-(p-Coumaroyl) serotonin		PDGFR
	N-(p-Coumaroyl) Serotonin is a polyphenol isolated from the seeds of safflower. N-(p-Coumaroyl) serotonin has antioxidant, cardioprotective effects after ischemia and antitumor activity, it may be beneficial in improving...		PDGFR
TN1564	Delphinidin 3-glucoside chloride	Delphinidin-3-O-glucoside chloride	Apoptosis , EGFR
	Delphinidin 3-glucoside chloride (Delphinidin-3-O-glucoside chloride) is a dietary phenolic substance found in Hibiscus sabdariffa extracts. Delphinidin 3-glucoside chloride has antioxidant activity, induces pro-apoptoti...		Apoptosis , EGFR
T3921	Punicalagin		SARS-CoV , HBV
	Punicalagin is a major ellagitannin found in pomegranates that is reported to produce antioxidant, anti-inflammatory, and anticancer effects. It has been shown to prevent high-fat diet-induced obesity-associated accumula...		SARS-CoV , HBV
TN1141	Isodeoxyelephantopin		NF-κB , Reactive Oxygen Species , Autophagy
	Isodeoxyelephantopin exerts antitumor effects on several cancer cells by inducing apoptosis , cell cycle arrest , and inhibiting proliferation. It enhances apoptosis and inhibit invasion and osteoclastogenesis by inhibit...		NF-κB , Reactive Oxygen Species , Autophagy
TN3284	8-Hydroxyodoroside A		Others
	An antitumor agent containing at least one compound selected from the group consisting of nerigoside, oleandrigenin, sarmentoside, oleaside A, oleandrin, 8β-hydroxy odoroside A, narciclasine, trans-dihydronarciclasine an...		Others
TN4421	Latisxanthone C		Others
	Latisxanthone C shows inhibitory effects on Epstein-Barr virus early antigen (EBV-EA) activation induced by 12-O-tetradecanoylphorbol-13-acetate (TPA) in Raji cells, it may be a valuable antitumor promoter.		Others
TN3019	4,9-Dihydroxy-alpha-lapachone		Others
	4,9-Dihydroxy-alpha-lapachone has antitumor-promoting effects, it exhibits significant inhibitory activity against 12-O-tetradecanoylphorbol 13-acetate (TPA)-induced Epstein-Barr virus early antigen (EBV-EA) activation i...		Others
TN4064	Flavoglaucin		Phosphatase , IL Receptor , TNF , NOS , NF-κB , COX , Nrf2 , Prostaglandin Receptor , Autophagy
	Flavoglaucin exhibits significant inhibitory effects on PTP1B, the IC50 value of 13.4, micrometer; it also shows good binding affinity for human opioid or cannabinoid receptors. Flavoglaucin appears to be an antitumor pr...
TN5233	Villosin		Others
	Villosin exhibits potent cytotoxic activity , it may be used as a potential lead molecule for antitumor therapeutic development. Villosin shows inhibitory effects against nitric oxide production in LPS and IFN-γ-induced ...		Others
T36303	Psammaplin A
	Psammaplin A, a marine metabolite, functions as a robust inhibitor of HDAC and DNA methyltransferases, displaying notable potency and selectivity as a DAC1 inhibitor, with an IC50 value of 0.9 nM. It exhibits antimicrobi...
TN2217	Sophoflavescenol		Others , Beta-Secretase , BACE , PDE , AChR , AChE
	Sophoflavescenol is a mixed inhibitor of PDE5 with a K(i) value of 0.005 microM. Sophoflavescenol has antioxidant, anti-inflammatory, and apoptotic effects , these effects might contribute to the antitumor activity witho...		Others , Beta-Secretase , BACE , PDE , AChR , AChE
TN2191	Scutebarbatine A		BCL , Caspase
	Scutebarbatine A shows significant antitumor effects on A549 cells in vivo and in vitro via mitochondria-mediated apoptosis by up-regulating expressions of caspase-3 and 9, and down-regulating Bcl-2. Scutebarbatine A and...		BCL , Caspase
T75520	Aplyronine A
	Aplyronine A, an actin-depolymerizing agent, exhibits antitumor and apoptosis effects. It is valuable in cancer research and studies on muscle contraction, cell motility, and cell division [1].
T83459	11α-O-Tigloyl-12β-O-acetyltenacigenin B		Aurora Kinase
	11α-O-Tigloyl-12β-O-acetyltenacigenin B, an ester derivative isolated from Garcinia cambogia (MTC), modulates the antitumor effects of Aurora-A in lymphoma through its parent compound, Tenacigenin B.		Aurora Kinase
TN5578	Abieta-8,11,13-triene-7,15,18-triol
	Abieta-8,11,13-triene-7alpha,15,18-triol,7alpha,8alpha,13beta,14beta-diepoxyabietan-18-oic acid, and 18-nor-abieta-8,11,13-triene-4alpha,7alpha,15-triol may have inhibitory effects on Epstein-Barr virus early antigen (EB...
T80777	Withaphysalin R
	Withaphysalin R (compound 5), a withanolide derived from the Solanaceae family, possesses an ergosterol-based steroid ester structure. This compound exhibits notable activities such as cytotoxic, immunosuppressive, antit...
TN2945	3-Hydroxybakuchiol		ATPase , Caspase
	3-Hydroxybakuchiol exerts cytotoxic and anti-proliferative effects on the TA3/Ha mouse mammary adenocarcinoma cell line and induces a decrease in the mitochondrial transmembrane potential, the activation of caspase-3, th...		ATPase , Caspase
T8291	2-Carene		Others
	2-Carene is a naturally occurring bicyclic monoterpene found in many essential oils such as pine, cedar and cypress. It has been found to have anti-inflammatory, antifungal and antibacterial activities, as well as antiox...		Others
T5157	9,13-Epidioxy-8(14)-abieten-18-oic acid		Others
	9,13β-Epidioxy-8(14)-abieten-18-oic acid has anti-inflammatory activities, it exhibits moderate activities on NO levels in LPS-stimulated murine microglia BV2 cells, with IC50 values of 57.3 ± 0.2 uM. It is also a potent...		Others
TN3616	Cedrelone		Apoptosis , MMP , Antifection
	Cedrelone is a citrulline analog and a phenazine biosynthesis-like domain protein (PBLD) activator.Cedrelone induces apoptosis in cancer cells.Cedrelone is a very potent inducer of apoptosis, causing cell cycle arrest.Ce...		Apoptosis , MMP , Antifection

天然物製品

Salvigenin

TMS1743

Synonym:

Target: MAO, Autophagy, ROS Kinase

Girinimbine

TN6097

Synonym: Girinimbin

Target: Apoptosis, Antioxidant, Antibacterial

Synonym: gamma Tocotrienol,gammaTocotrienol,gamma-Tocotrienol,D-gamma-Tocotrienol,Plastochromanol

Synonym: Mulberrochromene

Target: NF-κB, Antibacterial, STAT

(Z)-Butylidenephthalide

TN2326

Synonym: (Z)-3-Butylidenephthalide

Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Antibacterial

Hypocrellin A

T5771

Synonym:

Target: Antibacterial, PKC, Parasite

Syringin

T3408

Synonym: Lilacin,Syringoside,eleutheroside-b,Methoxyconiferine

Target: NOS, Autophagy

Kaempferitrin

T3386

Synonym: Lespedin,Kaempferol,Lespenephryl,Lespenefril,Kaempferol 3,7-dirhamnoside

Target: cell cycle arrest, Glucokinase, IGF-1R

Psoralenoside

TN1008

Synonym:

Target: CaMK, Calcium Channel, Histamine Receptor

Synonym: Allylglucosinolate,2-Propenylglucosinolate

Target: Others, Antioxidant

Chelerythrine

T6S0052

Synonym: Toddalin,Broussonpapyrine,Cheleritrine

Target: Apoptosis, BCL, PKC, Autophagy

2-Amino-2-dichlorobenzophenone

Target: Apoptosis, HIV Protease

Synonym: Bellidifoline,Bellidifolium

Target: Others, HIV Protease

N-(p-Coumaroyl) serotonin

TN1969

Synonym:

Target: PDGFR

Delphinidin 3-glucoside chloride

TN1564

Synonym: Delphinidin-3-O-glucoside chloride

Target: Apoptosis, EGFR

Punicalagin

T3921

Synonym:

Target: SARS-CoV, HBV

Isodeoxyelephantopin

TN1141

Synonym:

Target: NF-κB, Reactive Oxygen Species, Autophagy

4,9-Dihydroxy-alpha-lapachone

Target: Phosphatase, IL Receptor, TNF, NOS, NF-κB, COX, Nrf2, Prostaglandin Receptor, Autophagy

Target: Others, Beta-Secretase, BACE, PDE, AChR, AChE

11α-O-Tigloyl-12β-O-acetyltenacigenin B

T83459

Synonym:

Target: Aurora Kinase

Abieta-8,11,13-triene-7,15,18-triol

Target: ATPase, Caspase

9,13-Epidioxy-8(14)-abieten-18-oic acid

Target: Apoptosis, MMP, Antifection

Recombinant Proteins

Species：

Expression System：

Tag：

カタログ番号	製品名	Species	Expression System
TMPY-06983	IFN gamma Protein, Human, Recombinant (E. coli)	Human	E. coli
	IFN gamma, also known as IFNG, is a secreted protein that belongs to the type II interferon family. IFN gamma is produced predominantly by natural killer and natural killer T cells as part of the innate immune response, ...
TMPH-02451	IFN gamma Protein, Marmota monax, Recombinant (His)	Marmota monax	P. pastoris (Yeast)
	Produced by lymphocytes activated by specific antigens or mitogens. IFN-gamma, in addition to having antiviral activity, has important immunoregulatory functions. It is a potent activator of macrophages, it has antiproli...
TMPH-00373	IFN gamma Protein, Chicken, Recombinant (GST)	Chicken	E. coli
	Produced by lymphocytes activated by specific antigens or mitogens. IFN-gamma, in addition to having antiviral activity, has important immunoregulatory functions. It is a potent activator of macrophages, it has antiproli...
TMPK-00249	TRAIL R4/TNFRSF10D Protein, Human, Recombinant (His & Avi), Biotinylated	Human	HEK293 Cells
	TNF-related apoptosis inducing ligand (TRAIL) is a potential antitumor protein known for its ability to selectively eliminate various types of tumor cells without exerting toxic effects in normal cells and tissues. TRAIL...
TMPK-00248	TRAIL R4/TNFRSF10D Protein, Human, Recombinant (His & Avi)	Human	HEK293 Cells
	TNF-related apoptosis inducing ligand (TRAIL) is a potential antitumor protein known for its ability to selectively eliminate various types of tumor cells without exerting toxic effects in normal cells and tissues. TRAIL...

IFN gamma Protein, Human, Recombinant (E. coli)

TMPY-06983

Species: Human

Expression System: E. coli

IFN gamma Protein, Marmota monax, Recombinant (His)

TMPH-02451

Species: Marmota monax

Expression System: P. pastoris (Yeast)

IFN gamma Protein, Chicken, Recombinant (GST)

TMPH-00373

Species: Chicken

Expression System: E. coli

TRAIL R4/TNFRSF10D Protein, Human, Recombinant (His & Avi), Biotinylated

TMPK-00249

Species: Human

Expression System: HEK293 Cells

TRAIL R4/TNFRSF10D Protein, Human, Recombinant (His & Avi)

TMPK-00248

Species: Human

Expression System: HEK293 Cells

カタログ番号	製品名
L2152	Targeted Therapy Drug Library	119 compounds
	119 tumor-targeted drugs that can be used for high-throughput and high-content screening.
L6140	Saccharide and Glycoside Natural Product Library	595 compounds
	A unique collection of 595 saccharides and glycosides compounds can be used for HTS and HCS；
L9300	Macrocyclic Compound Library	210 compounds
	210 macrocyclic compounds of known activity for high-throughput, high-content screening;

ライブラリー

Targeted Therapy Drug Library

L2152

Compounds: 119

Saccharide and Glycoside Natural Product Library

L6140

Compounds: 595

Macrocyclic Compound Library

L9300

Compounds: 210